Title:
卵胞刺激ホルモン活性のアゴニスト
Document Type and Number:
Japanese Patent JP2004505051
Kind Code:
A
Abstract:
In one aspect, the present invention provides novel compounds. In addition, the invention provides a FSH receptor agonist, wherein the agonist binds to a FSH receptor having a FSH binding site and, wherein the agonist is noncompetitve with FSH for the FSH binding site. In another aspect, the invention provides methods of using the compounds of the present invention for diverse pharmaceutical applications including, for example, CNS antiischemic agents, agents with antipsychotic or other psychoactive properties, antimicrobial agents and mammalian fertility regulating agent.
Inventors:
Shore Man, Randall, A.
Janowski, Stephen, Dee.
Holmes, Christopher, Pee.
McLean, Derek
Roland, Beatrice
Barrett, Ronald, W.
Robert, Jay, Yi.
Wenlin, Khao
Gopal Sammy, Ariamara
Sam, Fuku-Wa
Huh, By Hua
Rogers, John, F.
Jetter, James, W.
Janowski, Stephen, Dee.
Holmes, Christopher, Pee.
McLean, Derek
Roland, Beatrice
Barrett, Ronald, W.
Robert, Jay, Yi.
Wenlin, Khao
Gopal Sammy, Ariamara
Sam, Fuku-Wa
Huh, By Hua
Rogers, John, F.
Jetter, James, W.
Application Number:
JP2002515259A
Publication Date:
February 19, 2004
Filing Date:
July 24, 2001
Export Citation:
Assignee:
SmithKline Beechham Corporation
International Classes:
A61K31/426; A61K31/427; A61K31/433; A61K31/4439; A61K31/5377; A61P5/10; A61P9/10; A61P15/00; A61P15/08; A61P25/18; A61P25/28; A61P31/00; A61P43/00; C07D277/14; C07D277/20; C07D417/02; C07D417/04; C07D417/06; C07D417/10; C07D417/12; C07D417/14; (IPC1-7): C07D277/14; A61K31/426; A61K31/427; A61K31/433; A61K31/4439; A61K31/5377; A61P5/10; A61P9/10; A61P15/00; A61P15/08; A61P25/18; A61P25/28; A61P31/00; A61P43/00; C07D417/02; C07D417/04; C07D417/06; C07D417/12; C07D417/14
Attorney, Agent or Firm:
Yusuke Hiraki
Satoshi Fujita
Ishii Teiji
Satoshi Fujita
Ishii Teiji