Title:
ピペラジニル-2(3H)-ベンゾキサゾロン化合物の経皮イオントフォレーシス送達
Document Type and Number:
Japanese Patent JP2007530512
Kind Code:
A
Abstract:
The present invention is related to the use of a compound of the general formula wherein R is methyl, ethyl, ethyl substituted with one or more fluorine atoms, or cycloalkyl-(C3-C7)-methyl optionally substituted with one or more fluorine atoms or benzyl optionally substituted with a group selected from phenyl, furanyl and thienyl which groups are optionally substituted with 1-3 substituents from the group hydroxy, halogen, C1-4-alkoxy, C1-4-alkyl, cyano, aminocarbonyl, mono- or di-C1-4-alkylaminocarbonyl; and pharmaceutically acceptable salts and prodrugs thereof, for the manufacture of a composition for transdermal administration by iontophoresis.
Inventors:
Boostra, Johanna A
Van den berg, daleck-yan
Bellburn, Frederik Jei
Congee Balam, Likemar Buoy
Bunga, Kay Kay
Vemura Paris, Biswati
Van Schallenburg, JAM
Houendrik, Hendrik
Van den berg, daleck-yan
Bellburn, Frederik Jei
Congee Balam, Likemar Buoy
Bunga, Kay Kay
Vemura Paris, Biswati
Van Schallenburg, JAM
Houendrik, Hendrik
Application Number:
JP2007504423A
Publication Date:
November 01, 2007
Filing Date:
March 25, 2005
Export Citation:
Assignee:
Solvay Pharmaceuticals B.V.
International Classes:
A61K31/496; A61K9/06; A61K9/08; A61K47/04; A61K47/12; A61N1/30; A61N1/32; A61P25/04; A61P25/14; A61P25/16
Domestic Patent References:
| JP2003532729A | 2003-11-05 | |||
| JP2003532676A | 2003-11-05 |
Foreign References:
| WO2003068207A2 | 2003-08-21 | |||
| US20040013620A1 | 2004-01-22 | |||
| EP0529510A1 | 1993-03-03 |
Attorney, Agent or Firm:
Heikichi Odashima