縮合2環系mTOR阻害剤 - OSI Pharmaceuticals Incorporated

Title:

縮合2環系mTOR阻害剤

Document Type and Number:

Japanese Patent JP2009519222

Kind Code:

A

Abstract:

A compound represented by the formula I or II:

Inventors:

Chiyoung, Shin
Coat, heather
Crew, Andrew-Filip
Don, Han-Chin
Ayako Honda
Marvi Hill, Mark Joseph
Tavares, Paula A.R.
One, Chin
Warner Douglas S
Marvi Hill, Kristen Michel
Shiyu, Cam Davryu
Panika, business
Baladwazi, Apuruba
Arnold, Lee Day
Chin, Maycheon
Brian Bourk
Won, Chinghua
Beard, The Ames David

Application Number:

JP2008541334A

Publication Date:

May 14, 2009

Filing Date:

November 15, 2006

Export Citation:

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Assignee:

OSI Pharmaceuticals Incorporated

International Classes:

C07D487/04; A61K31/519; A61K31/53; A61K45/00; A61K45/06; A61P9/10; A61P19/02; A61P25/00; A61P35/00; A61P37/02; A61P37/06; A61P43/00; C07D253/06; C07F5/02

Domestic Patent References:

JP4491510B2	2010-06-30
JP2009514882A	2009-04-09
JP2008520744A	2008-06-19
JP4491510B2	2010-06-30

Foreign References:

WO2005037836A2	2005-04-28
WO2005047289A1	2005-05-26
WO2004056830A1	2004-07-08
WO2005097800A1	2005-10-20
WO2005037836A2	2005-04-28

Other References:

JPN6012035999; Ｂｉｓｈｏｐ，　Ａｎｔｈｏｎｙ　Ｃ．他: 'Ｇｅｎｅｒａｔｉｏｎ　ｏｆ　Ｍｏｎｏｓｐｅｃｉｆｉｃ　Ｎａｎｏｍｏｌａｒ　Ｔｙｒｏｓｉｎｅ　Ｋｉｎａｓｅ　Ｉｎｈｉｂｉｔｏｒｓ　ｖｉａ　ａ　　　　　Ｃｈｅｍｉｃａｌ　Ｇｅｎｅｔｉｃ　Ａｐｐｒｏａｃｈ' Ｊｏｕｒｎａｌ　ｏｆ　ｔｈｅ　Ａｍｅｒｉｃａｎ　Ｃｈｅｍｉｃａｌ　Ｓｏｃｉｅｔｙ１２１（４）, 1999, ６２７-６３１
JPN5008019280; ＢＥＲＧＳＴＲＯＭ　Ｄ: ＪＯＵＲＮＡＬ　ＯＦ　ＯＲＧＡＮＩＣ　ＣＨＥＭＩＳＴＲＹＶ５６　Ｎ１９, 1991, Ｐ５５９８-５６０２, ＡＭＥＲＩＣＡＮ　ＣＨＥＭＩＣＡＬ　ＳＯＣＩＥＴＹ
JPN6012035999; Ｂｉｓｈｏｐ，　Ａｎｔｈｏｎｙ　Ｃ．他: 'Ｇｅｎｅｒａｔｉｏｎ　ｏｆ　Ｍｏｎｏｓｐｅｃｉｆｉｃ　Ｎａｎｏｍｏｌａｒ　Ｔｙｒｏｓｉｎｅ　Ｋｉｎａｓｅ　Ｉｎｈｉｂｉｔｏｒｓ　ｖｉａ　ａ　　　　　Ｃｈｅｍｉｃａｌ　Ｇｅｎｅｔｉｃ　Ａｐｐｒｏａｃｈ' Ｊｏｕｒｎａｌ　ｏｆ　ｔｈｅ　Ａｍｅｒｉｃａｎ　Ｃｈｅｍｉｃａｌ　Ｓｏｃｉｅｔｙ１２１（４）, 1999, ６２７-６３１
JPN5008019280; ＢＥＲＧＳＴＲＯＭ　Ｄ: ＪＯＵＲＮＡＬ　ＯＦ　ＯＲＧＡＮＩＣ　ＣＨＥＭＩＳＴＲＹＶ５６　Ｎ１９, 1991, Ｐ５５９８-５６０２, ＡＭＥＲＩＣＡＮ　ＣＨＥＭＩＣＡＬ　ＳＯＣＩＥＴＹ

Attorney, Agent or Firm:

Yoshio Kawaguchi
Makoto Ono
Chihiro Watanabe
Kenkyo Kanayama
Katsuma Osaki
Mitsuaki Tsubokura

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