Title:
6-(ピペリジン-4-イルオキシ)-2H-イソキノリン-1-オン塩酸塩の多形体
Document Type and Number:
Japanese Patent JP2014518236
Kind Code:
A
Abstract:
The present invention relates to new crystalline polymorphs of 6-(Piperidin-4-yloxy)-2H-isoquinolin-1-one hydrochloride, processes for their preparation and their use, in particular for the preparation of medicaments.
Inventors:
Norbert Nagel
Bruno Baumgartner
Harald Berchtort
Oliver Plettenburg
Dieter Cardellite
Mandy Mornicke
Gimon Gesler
Joachim Tillner
Bruno Baumgartner
Harald Berchtort
Oliver Plettenburg
Dieter Cardellite
Mandy Mornicke
Gimon Gesler
Joachim Tillner
Application Number:
JP2014517676A
Publication Date:
July 28, 2014
Filing Date:
June 27, 2012
Export Citation:
Assignee:
SANOFI
International Classes:
C07D401/12; A61K31/4422; A61K31/4725; A61K45/00; A61P1/16; A61P3/00; A61P3/10; A61P7/02; A61P9/00; A61P9/04; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P11/08; A61P13/08; A61P13/12; A61P15/06; A61P15/10; A61P19/08; A61P25/00; A61P25/04; A61P25/28; A61P27/02; A61P27/06; A61P29/00; A61P31/04; A61P35/00; A61P37/06
Domestic Patent References:
| JP2003519698A | 2003-06-24 |
Foreign References:
| WO2008077550A1 | 2008-07-03 | |||
| WO2007012421A1 | 2007-02-01 | |||
| WO2009080335A1 | 2009-07-02 |
Other References:
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川口洋子ら: "医薬品と結晶多形", 生活工学研究, vol. 4, no. 2, JPN6014015069, 2002, pages 310 - 317, ISSN: 0003265264
"新医薬品の規格及び試験方法の設定について", 医薬審発第５６８号, JPN6010021254, 2001, ISSN: 0003265265
大島寛: "結晶多形・擬多形の析出挙動と制御", PHARM STAGE, vol. 6, no. 10, JPN6011001457, 15 January 2007 (2007-01-15), pages 48 - 53, ISSN: 0003265266
山野光久: "医薬品のプロセス研究における結晶多形現象への取り組み", 有機合成化学協会誌, vol. 65, no. 9, JPN6010003277, 1 September 2007 (2007-09-01), pages 907 - 69, ISSN: 0003265267
BYRN S: "PHARMACEUTICAL SOLIDS: A STRATEGIC APPROACH TO REGULATORY CONSIDERATIONS", PHARMACEUTICAL RESEARCH, vol. V12 N7, JPN5013009960, 1 July 1995 (1995-07-01), US, pages 945 - 954, XP055307460, ISSN: 0003265268, DOI: 10.1023/A:1016241927429
Attorney, Agent or Firm:
Junji Yuda
Noriyuki Takebayashi
Noriyuki Takebayashi