Title:
オキサゼチジン誘導体、それらの調製方法並びにヒト医療及び化粧品におけるそれらの使用
Document Type and Number:
Japanese Patent JP2014518238
Kind Code:
A
Abstract:
Compounds that are agonists of the MCIR receptor and that exhibit reduced toxicity relative to other compounds of the same class are described. These compounds can have the general formula (I) wherein: R1 represents a cyclopropylmethyl or a 4-hydroxybutyl group; R2 represents a hydrogen atom or a methyl group; and also the salts and enantiomers of the corresponding compounds of general formula (I). Also described, are methods for treating hypopigmentary pathologies and photosensitive dermatoses.
Inventors:
Clair Buix-Peter
Application Number:
JP2014517715A
Publication Date:
July 28, 2014
Filing Date:
June 28, 2012
Export Citation:
Assignee:
Galderma Research and Development
International Classes:
C07D403/12; A61K8/49; A61K31/4178; A61P1/04; A61P1/14; A61P1/16; A61P1/18; A61P3/04; A61P3/06; A61P7/02; A61P9/00; A61P9/10; A61P9/12; A61P11/00; A61P11/02; A61P11/06; A61P13/00; A61P13/10; A61P15/08; A61P15/10; A61P17/00; A61P17/06; A61P17/14; A61P19/02; A61P19/10; A61P21/00; A61P25/00; A61P25/08; A61P25/16; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P29/00; A61P31/04; A61P31/10; A61P31/12; A61P35/00; A61P37/06; A61P37/08; A61Q5/00; A61Q19/08
Domestic Patent References:
| JP2004532838A | 2004-10-28 | |||
| JP2007510717A | 2007-04-26 | |||
| JP2005511475A | 2005-04-28 | |||
| JP2004532838A | 2004-10-28 | |||
| JP2007510717A | 2007-04-26 | |||
| JP2005511475A | 2005-04-28 |
Foreign References:
| WO2010052255A1 | 2010-05-14 | |||
| WO2010052253A1 | 2010-05-14 | |||
| WO2010052253A1 | 2010-05-14 | |||
| WO2010052255A1 | 2010-05-14 |
Attorney, Agent or Firm:
Yasuhiko Murayama
Masatake Shiga
Takashi Watanabe
Shinya Mitsuhiro
Masatake Shiga
Takashi Watanabe
Shinya Mitsuhiro