Title:
オキシインドールジオキサン誘導体の合成において適当な中間体である化合物の合成法
Document Type and Number:
Japanese Patent JP5295103
Kind Code:
B2
Abstract:
The present invention provides methods for preparing compounds having activity as dopamine autoreceptor agonists and partial agonists at the postsynaptic dopamine D2 receptor. These compounds are useful for treating dopaminergic disorders, such as schizophrenia, schizoaffective disorder, Parkinson's disease, Tourette's syndrome, hyperprolactinemia, and drug addiction.
Inventors:
Rocco Jay Galante
Application Number:
JP2009512182A
Publication Date:
September 18, 2013
Filing Date:
May 25, 2007
Export Citation:
Assignee:
Weiss LRC
International Classes:
C07D319/20; C07D491/056; A61K31/407; A61P25/18
Domestic Patent References:
| JP9249671A |
Other References:
FORBES,I.T. et al,Synthesis, Biological Activity, and Molecular Modeling Studies of Selective 5-HT2C/2B Receptor Antagonists,Journal of Medicinal Chemistry,1996年,Vol.39, No.25,pp.4966-4977
Attorney, Agent or Firm:
Mitsuo Tanaka
Hiroshi Yamazaki
Kenji Tomita
Hiroshi Yamazaki
Kenji Tomita