置換ピロリジンアミド、それの製造方法、及び、それの薬剤としての使用

Japanese Patent JP5397959

B2

Substituted amide compounds (I) and their tautomers, enantiomers, diastereomers or salts, are new. Substituted amide compounds of formula (I) and their tautomers, enantiomers, diastereomers or salts, are new. D : a substituted bicyclic ring system; L-E-G-J : a C-C-C-C-group, which is optionally substituted by R 4> and R 5>; L 1>, L 2>C(O); R 4>e.g. H, 1-6C-alkyl, 2-6C-alkenyl or 2-6C-alkynyl; R 5>e.g. H, 1-5C-alkyl or 2-5C-alkenyl; and M : e.g. phenyl or pyridyl ring. With provisos. Full Definitions are given in the DEFINITIONS (Full Definitions) Field. [Image] ACTIVITY : Anticoagulant; Antiinflammatory; Vasotropic; Thrombolytic; Antibacterial; Immunosuppressive; Respiratory-Gen; Antiulcer; Gastrointestinal-Gen; Cardiant; Cerebroprotective; Neuroprotective; Nootropic; Antiparkinsonian; Cytostatic; Antiarthritic; Antirheumatic; Vulnerary. MECHANISM OF ACTION : Thrombosis factor Xa inhibitor; Serine protease inhibitor.

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Gerlach Kai
Prepke Henning
Wienen Wolfgang
Schuler-Mets Anette
Derman Georg
Na Herbert

JP2010500259A

January 22, 2014

March 26, 2008

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Boehringer Ingelheim International GmbH

C07D401/06; C07D401/14; C07D405/14; C07D409/14; C07D487/04; C07D495/04; C07D513/04; A61K31/404; A61K31/4365; A61K31/4725; A61K31/4985; A61K31/55; A61K31/551; A61P7/02; A61P9/00; A61P11/00; A61P19/02; A61P25/16; A61P25/28; A61P29/00; A61P35/00; A61P43/00; C07D403/06

JP2006520790A
JP2006510582A

WO2005032472A1
WO2004082687A1
WO2004017908A1
WO2003099276A1
WO2002014308A1

Sadao Kumakura
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Kobayashi Machiko

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