Title:
抹消性ＮＭＤＡ受容体アンタゴニストとしての新規なジゾシルピン誘導体
Document Type and Number:
Japanese Patent JP6827665
Kind Code:
B2
Abstract:
The present invention relates to compounds of formula (I):for use as peripheral NMDA receptor antagonists.
Inventors:
Cohen-Kaminsky, Sylvia
Hambert, mark
Dumas, Sebastian
Bull-Merche, Jill
Messa Woody, Samir
Brion, Jean-Daniel
Arami, Mouad
Jill Galvani
Hambert, mark
Dumas, Sebastian
Bull-Merche, Jill
Messa Woody, Samir
Brion, Jean-Daniel
Arami, Mouad
Jill Galvani
Application Number:
JP2019517168A
Publication Date:
February 10, 2021
Filing Date:
June 13, 2017
Export Citation:
Assignee:
Anstitut National de la Sant'Edela Recherche Medical (Anselm)
Center National de la Recherche Scientific
INSTITUT GUSTAVE-ROUSSY
Assistance Public-Hopiteau de Paris
Hospital Marie Run Long
Center National de la Recherche Scientific
INSTITUT GUSTAVE-ROUSSY
Assistance Public-Hopiteau de Paris
Hospital Marie Run Long
International Classes:
C07D451/00; A61K31/4748; A61K45/00; A61P3/10; A61P7/00; A61P9/10; A61P9/12; A61P11/00; A61P13/12; A61P17/00; A61P17/06; A61P19/10; A61P25/04; A61P29/00; A61P31/00; A61P35/00; A61P37/02; A61P37/08; A61P43/00
Domestic Patent References:
| JP9216882A |
Other References:
LINDERS, J. T. M. et al.,Letters in Drug Design & Discovery,2010年,Vol. 7,pp. 79-87
THOMPSON, W. J. et al.,Journal of Medicinal Chemistry,1990年,Vol. 33,pp. 789-808
ELHALLAOUI, M. et al.,Internationial Journal of Molecular Sciences,2003年,Vol. 4,pp. 249-262
THOMPSON, W. J. et al.,Journal of Medicinal Chemistry,1990年,Vol. 33,pp. 789-808
ELHALLAOUI, M. et al.,Internationial Journal of Molecular Sciences,2003年,Vol. 4,pp. 249-262
Attorney, Agent or Firm:
Mitsuo Matsui