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Title:
【発明の名称】サイクロスポリン誘導体含有医薬組成物
Document Type and Number:
Japanese Patent JPH07505872
Kind Code:
A
Abstract:
A pharmaceutical composition containing ([3'-desoxy-3'-oxo-MeBmt]<1>-[Val]<2>-Ciclosporin) as an active ingredient. The composition is formulated as a microemulsion or microemulstion preconcentrate using a carrier medium comprising a hydrophilic phase; a transesterified ethoxylated vegetable oil; and a surfactant. The composition has good stability and biopharmaceutical properties and is useful in the treatment of multiple drug resistance syndrome in humans.

Inventors:
Mainzer, Armin
Richter, Friedrich
Vondersche, Jackie Francis
Application Number:
JP51799893A
Publication Date:
June 29, 1995
Filing Date:
April 20, 1993
Export Citation:
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Assignee:
Novartis Actien Gezel Shaft
International Classes:
A61K9/107; A61K38/00; A61K38/13; A61K47/14; A61K47/44; (IPC1-7): A61K38/00; A61K9/107
Domestic Patent References:
JPH02121929A1990-05-09
JPS6445396A1989-02-17
JPS54132223A1979-10-15
Attorney, Agent or Firm:
Aoyama Ryo (1 person outside)



 
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