Title:
COMPOUNDS AND METHODS FOR TARGETED DEGRADATION OF THE ANDROGEN RECEPTOR
Document Type and Number:
Japanese Patent JP2023040072
Kind Code:
A
Abstract:
To provide bifunctional compounds which find utility to degrade and inhibit Androgen Receptor.SOLUTION: There is provided a compound represented by following formula (example 1).SELECTED DRAWING: Figure 1
Inventors:
Jin Mae Chung
Crew Andrew Pea.
Don Hankin
Wang Jin
Ferraro Caterina
Chen Chin
Chien Yimin
Crew Andrew Pea.
Don Hankin
Wang Jin
Ferraro Caterina
Chen Chin
Chien Yimin
Application Number:
JP2022206686A
Publication Date:
March 22, 2023
Filing Date:
December 23, 2022
Export Citation:
Assignee:
ARVINAS OPERATIONS, INC.
International Classes:
C07D233/86; A61K45/00; A61K47/66; A61P25/02; A61P35/00; A61P43/00; C07C255/54; C07D213/82; C07D231/14; C07D235/02; C07D237/24; C07D239/42; C07D241/28; C07D401/04; C07D401/10; C07D403/10; C07D403/14; C07D413/14; C07D419/10; C07D419/14; C07D471/10; C07D491/107
Attorney, Agent or Firm:
Shimizu Hatsushi
Masao Haruna
Hirotaka Yamaguchi
Shun Jinbe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Hideki Kodera
Masato Ozeki
Kazuya Kawamoto
Masao Haruna
Hirotaka Yamaguchi
Shun Jinbe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Hideki Kodera
Masato Ozeki
Kazuya Kawamoto
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