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Title:
心不整脈および心不全の処置のための化合物
Document Type and Number:
Japanese Patent JP7359460
Kind Code:
B2
Abstract:
This disclosure concerns compounds and a method for modulating the activity of calcium ion channels, including Ca2+-induced (or Ca2+-activated) calcium release channels and conformationally coupled calcium release channels such as ryanodine receptors. Some of the compounds have a structure according to formula I, or a stereoisomer, tautomer, hydrate, solvate, prodrug, or pharmaceutically acceptable salt thereof.

Inventors:
Cibrian Vasquez, Marta
Taina Schmutz, Joseph Rajan
boatman, douglas
Application Number:
JP2021502722A
Publication Date:
October 11, 2023
Filing Date:
March 28, 2019
Export Citation:
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Assignee:
Elex Biotech, Inc.
International Classes:
C07C217/84; A61K31/136; A61K31/185; A61K31/4035; A61K31/41; A61K31/416; A61K31/4245; A61P9/10; A61P43/00; C07C309/24; C07D231/56; C07D257/04; C07D271/06
Domestic Patent References:
JP2009526072A
JP2010529029A
JP2004515518A
Foreign References:
WO2008061109A2
Other References:
REGISTRY(STN)[online],2016年08月03日,[検索日2023.01.19], CAS登録番号1966110-41-7など
REGISTRY(STN)[online],2016年06月13日,[検索日2023.01.19], CAS登録番号 1930380-26-9など
Attorney, Agent or Firm:
Shusaku Yamamoto
Natsuki Morishita
Takatoshi Iida
Daisuke Ishikawa
Kensaku Yamamoto