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Title:
線維芽細胞活性化タンパク質の阻害剤
Document Type and Number:
Japanese Patent JP2021506972
Kind Code:
A
Abstract:
線維芽細胞活性化タンパク質(FAP)を調節するための化合物および組成物が記載されている。本化合物および組成物は、過増殖性疾患を含む疾患の治療のための治療剤としての使用を見出し得る。【選択図】図6C

Inventors:
Alfaro, Jennifer
Bellmawr, Sebastian
Bernares, Sebastian
Pujara, Brahman
Panpatil, Dayanando
Bat, Berwana
Application Number:
JP2020552675A
Publication Date:
February 22, 2021
Filing Date:
December 14, 2018
Export Citation:
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Assignee:
Praxis Biotech LLC
International Classes:
C07D207/16; A61K31/216; A61K31/40; A61K31/4025; A61K31/403; A61K31/416; A61K31/422; A61K31/4439; A61K31/4545; A61K31/4709; A61K31/4725; A61K31/517; A61K31/5377; A61K31/55; A61K45/00; A61P1/04; A61P3/04; A61P7/00; A61P9/10; A61P11/00; A61P17/02; A61P19/02; A61P29/00; A61P35/00; A61P43/00; C07D401/12; C07D401/14; C07D403/12; C07D405/12; C07D405/14; C07D413/14; C07D471/04; C07D487/04; C07D491/048
Domestic Patent References:
JP2009507011A2009-02-19
Foreign References:
WO2017189569A12017-11-02
Other References:
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 22, no. 10, JPN6022050808, 2012, pages 3412 - 3417, ISSN: 0004937785
JOURNAL OF MEDICINAL CHEMISTRY, vol. 57, no. 7, JPN6022050807, 2014, pages 3053 - 3074, ISSN: 0004937786
Attorney, Agent or Firm:
Hiraki International Patent Office