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Title:
ホスホジエステラーゼ7に対するピリミジン阻害剤
Document Type and Number:
Japanese Patent JP2005500294
Kind Code:
A
Abstract:
Pyrimidine phosphodiesterase 7 (PDE 7) inhibitors of the following formula wherein R1, R2, Z, J and L are described herein, and analogs thereof are provided which are useful in treating T-cell mediated diseases.

Inventors:
Guo Junkin
Joseph Barbosa
William John Pitts
Marianne Karlsen
Claude Quesnel
Marco Dodier
Application Number:
JP2003504902A
Publication Date:
January 06, 2005
Filing Date:
June 17, 2002
Export Citation:
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Assignee:
BRISTOL-MYERS SQUIBB COMPANY
International Classes:
A61K31/00; A61K31/496; A61K31/505; A61K31/506; A61K31/513; A61K31/517; A61K31/519; A61K31/522; A61K31/538; A61K31/5513; A61K45/00; A61P1/00; A61P1/04; A61P3/10; A61P5/14; A61P9/10; A61P11/00; A61P11/04; A61P11/06; C07D491/113; A61P17/04; A61P17/06; A61P17/14; A61P19/00; A61P19/02; A61P21/04; A61P25/00; A61P25/28; A61P29/00; A61P35/00; A61P37/00; A61P37/06; A61P43/00; C07D403/12; C07D417/12; C07D417/14; C07D471/04; C07D473/00; C07D473/16; C07D487/04; C07D491/10; C07D498/10; (IPC1-7): C07D417/12; A61K31/496; A61K31/506; A61K31/538; A61K31/5513; A61K45/00; A61P1/00; A61P3/10; A61P9/10; A61P11/06; A61P17/06; A61P25/00; A61P29/00; A61P37/06; A61P43/00; C07D403/12; C07D417/14; C07D491/113; C07D498/10
Attorney, Agent or Firm:
Kyousei Tamura
Nagatoshi Shinagawa