THIENO-(1,3)-OXAZIN-4-ONES WITH LIPASE INHIBITING ACTIVITY

Japanese Patent JP2010159260

A

To provide a compound for treating obesity or obesity-related disorders.

The compound of formula (I) (wherein A is an optionally substituted thienyl moiety; Y is O, S or NR2; R1is a branched or unbranched alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, aryl, arylalkyl, reduced arylalkyl, arylalkenyl, heteroaryl, heteroarylalkyl, heteroarylalkenyl, reduced aryl, reduced heteroaryl, reduced heteroarylalkyl or a substituted derivative of any of the above groups; and R2is hydrogen or a group as defined for R1) or a pharmaceutically acceptable salt, ester, amide or prodrug thereof is described.

COPYRIGHT: (C)2010,JPO&INPIT

WO/2002/078616	METHODS FOR INCREASING SEROTONIN LEVELS BY ADMINISTERING (-)-HYDROXYCITRIC ACID
JP2004105176	FUNCTIONAL FOOD AND MEDICAMENT CONTAINING BRASSICA CAMPESTRIS OR ITS HYBRID AND HAVING EFFECT OF DECREASING BLOOD GLUCOSE
WO/2002/015887	CONSUMABLE CONTAINER

HODSON HAROLD FRANCIS
DUNK CHRISTOPHER ROBERT
PALMER RICHARD MICHAEL JOHN
MITCHELL DALE ROBERT
BIRAULT VERONIQUE
HUNT RUSSELL GEORGE

JP2010019160A

July 22, 2010

January 29, 2010

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NORGINE BV

A23L1/30; A23L3/3544; C07D498/04; A61K8/49; A61K31/4365; A61K31/535; A61K31/5365; A61P1/00; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/12; A61P25/00; A61P43/00; A61Q19/10; C07D498/14; C11D3/28; C11D3/48; C12N9/99

JP2005518383A	2005-06-23
JP2005527469A	2005-09-15

WO2001018181A2	2001-03-15
WO2000040247A1	2000-07-13
WO2000040569A1	2000-07-13
WO2001053278A1	2001-07-26

Takehiko Suzue
Kurata Masatoshi
Satoshi Kono
Makoto Nakamura
Yoshihiro Fukuhara
Takashi Mine
Toshio Shirane
Sadao Muramatsu
Nobuhisa Nogawa
Kocho Chojiro
Naoki Kono
Katsu Sunagawa
Katsumura Hiro
Tatsushi Sato
Takashi Okada
Mihoko Horiuchi
Takenori Masanori
Takuzo Ichihara
Yamashita Gen

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