Title:
ALKENE MIMICS
Document Type and Number:
WIPO Patent Application WO2006020417
Kind Code:
A3
Abstract:
Ac-Phe-Tyr-phosphoSer-?[CH=C]-Pro-Arg-NH2AND Fmoc-bis(pivaloylmethoxy)phosphoSer-?[CH=C]-Pro-2-aminoethyl-(3-indole); and their Phospho-(D)-serine stereoisomers are novel compounds. ? refers to a pseudo amide. Such novel compounds advantageously may be used as alkene mimics.
Inventors:
ETZKORN FELCIA A (US)
WANG XIAODONG X (US)
XU BAILING (US)
WANG XIAODONG X (US)
XU BAILING (US)
Application Number:
PCT/US2005/026821
Publication Date:
July 13, 2006
Filing Date:
July 29, 2005
Export Citation:
Assignee:
VIRGINIA TECH INTELL PROP (US)
ETZKORN FELCIA A (US)
WANG XIAODONG X (US)
XU BAILING (US)
ETZKORN FELCIA A (US)
WANG XIAODONG X (US)
XU BAILING (US)
International Classes:
A61K31/405; C07F9/06
Other References:
DATABASE CAPLUS [online] ZHANG ET AL.: "Inhibitors Targeting the Enzymatic Activity and Biological Function of Pin1", XP003000987, accession no. STN Database accession no. (2004:755045)
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