ANDROGEN RECEPTOR MODULATING COMPOUNDS

Title:

ANDROGEN RECEPTOR MODULATING COMPOUNDS

Document Type and Number:

WIPO Patent Application WO/2011/051540

Kind Code:

A8

Abstract:

Compounds of formula (I) wherein R1 to R16, A. B and E are as defined in the claims and pharmaceutically acceptable salts and esters thereof, are disclosed. The compounds of formula (I) possess utility as tissue-selective androgen receptor modulators (SARM) and are particularly useful as medicaments in the treatment of prostate cancer and other AR dependent conditions and diseases where AR antagonism is desired.

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Inventors:

WOHLFAHRT GERD (FI)
TOERMAEKANGAS OLLI (FI)
SALO HARRI (FI)
HOEGLUND IISA (FI)
KARJALAINEN ARJA (FI)
KNUUTTILA PIA (FI)
HOLM PATRIK (FI)
RASKU SIRPA (FI)
VESALAINEN ANNIINA (FI)

Application Number:

PCT/FI2010/000065

Publication Date:

May 24, 2012

Filing Date:

October 27, 2010

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Assignee:

ORION CORP (FI)
WOHLFAHRT GERD (FI)
TOERMAEKANGAS OLLI (FI)
SALO HARRI (FI)
HOEGLUND IISA (FI)
KARJALAINEN ARJA (FI)
KNUUTTILA PIA (FI)
HOLM PATRIK (FI)
RASKU SIRPA (FI)
VESALAINEN ANNIINA (FI)

International Classes:

C07D231/14; A61K31/416; A61K31/42; A61K31/438; A61K31/44; A61K31/4523; A61K31/497; A61K31/5377; A61P35/00; C07D401/12; C07D403/12; C07D405/12; C07D413/12; C07D417/12

Attorney, Agent or Firm:

ORION CORPORATION (Espoo, FI)

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