Title:
CARBOXYLIC ACID DERIVATIVES AND ADHESION MOLECULE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT
Document Type and Number:
WIPO Patent Application WO/2001/007400
Kind Code:
A1
Abstract:
Substances inhibiting cell adhesion mediated by adhesion molecules (in particular, VLA-4) which enable the prevention and treatment of inflammatory diseases caused by leukocyte (for example, monocyte, lymphocyte or eosinocyte) infiltration. A group of carboxylic acid derivatives exemplified by a compound represented by the formula (140) and adhesion molecule inhibitors containing the same as the active ingredient
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Inventors:
TAKAHASHI TOSHIYA (JP)
TAKANO YOSHIO (JP)
ISHIGAKI TAKESHI (JP)
FUNAHASHI MIYUKI (JP)
KANEKO MASAYUKI (JP)
KAINOH MIE (JP)
TAKANO YOSHIO (JP)
ISHIGAKI TAKESHI (JP)
FUNAHASHI MIYUKI (JP)
KANEKO MASAYUKI (JP)
KAINOH MIE (JP)
Application Number:
PCT/JP2000/004965
Publication Date:
February 01, 2001
Filing Date:
July 26, 2000
Export Citation:
Assignee:
TORAY INDUSTRIES (JP)
TAKAHASHI TOSHIYA (JP)
TAKANO YOSHIO (JP)
ISHIGAKI TAKESHI (JP)
FUNAHASHI MIYUKI (JP)
KANEKO MASAYUKI (JP)
KAINOH MIE (JP)
TAKAHASHI TOSHIYA (JP)
TAKANO YOSHIO (JP)
ISHIGAKI TAKESHI (JP)
FUNAHASHI MIYUKI (JP)
KANEKO MASAYUKI (JP)
KAINOH MIE (JP)
International Classes:
A61P29/00; A61P43/00; C07C229/22; C07C229/36; C07C233/22; C07C233/47; C07C233/51; C07C233/83; C07C233/87; C07C235/12; C07C235/34; C07C235/52; C07C235/60; C07C237/12; C07C237/22; C07C251/24; C07C271/22; C07C275/28; C07C275/30; C07C275/42; C07C311/21; C07C323/59; C07D207/08; C07D239/46; C07K5/02; C07K5/06; C07K5/078; C07K5/097; A61K38/00; (IPC1-7): C07C233/51; A61K31/198; A61K31/216; A61K31/22; A61K31/222; A61K31/235; A61K31/27; A61K31/277; A61K31/40; A61K31/505; A61K38/00; A61P29/00; A61P43/00; C07C233/87; C07C235/12; C07C235/66; C07C237/22; C07C275/42; C07C311/21; C07C323/59; C07C329/06; C07D207/08; C07D239/47; C07K5/062
Domestic Patent References:
WO1996022966A1 | 1996-08-01 |
Attorney, Agent or Firm:
Tanigawa, Hidejiro (Patent Firm 6F Iwata Bldg. 5-1, Iidabashi 4-chome Chiyoda-ku Tokyo, JP)
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