Title:
HETEROCYCLES AS MODULATORS OF NSD ACTIVITY
Document Type and Number:
WIPO Patent Application WO/2024/073282
Kind Code:
A3
Abstract:
Disclosed herein are amino bicyclic nitrogen heterocyclic ring system compounds which inhibit nuclear receptor-binding SET domain proteins (NSD's), such as 6-amino-9H-purin-9-yl, imidazo[2,1-f][1,2,4]triazin-4-amine, 4-amino pyrazolo[1,5-a][1,3,5]triazin-8-yl ring systems, and in particular the 8-amino imidazo[1,2-a]pyrazin-3-yl system, as well as their pharmaceutical formulations, and their methods of utilization in the treatment of NSD-mediated diseases, such as certain cancers.
Inventors:
LE KANG (US)
SOTH MICHAEL (US)
HAMILTON MATTHEW (US)
RAMASWAMY SUYAMBU KESAVA VIJAYAN (US)
JONES PHILIP (US)
SOTH MICHAEL (US)
HAMILTON MATTHEW (US)
RAMASWAMY SUYAMBU KESAVA VIJAYAN (US)
JONES PHILIP (US)
Application Number:
PCT/US2023/074671
Publication Date:
May 16, 2024
Filing Date:
September 20, 2023
Export Citation:
Assignee:
UNIV TEXAS (US)
International Classes:
A61K31/4985; C07D487/04
Attorney, Agent or Firm:
STEVENS, Lauren (US)
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