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Title:
HETEROCYCLIC COMPOUND
Document Type and Number:
WIPO Patent Application WO/2015/002231
Kind Code:
A1
Abstract:
The present invention relates to compounds (I), which have RORγt inhibitory effects, and salts thereof. In formula (I), each notation is as described in the Specification. (I)

Inventors:
YAMAMOTO SATOSHI (JP)
SHIRAI JUNYA (JP)
WATANABE HIROYUKI (JP)
FUKUMOTO SHOJI (JP)
ODA TSUNEO (JP)
TOKUHARA HIDEKAZU (JP)
TOMATA YOSHIHIDE (JP)
ISHII NAOKI (JP)
TAWADA MICHIKO (JP)
KOUNO MITSUNORI (JP)
OCHIDA ATSUKO (JP)
IMADA TAKASHI (JP)
FUKASE YOSHIYUKI (US)
YUKAWA TOMOYA (US)
Application Number:
PCT/JP2014/067650
Publication Date:
January 08, 2015
Filing Date:
July 02, 2014
Export Citation:
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Assignee:
TAKEDA PHARMACEUTICAL (JP)
International Classes:
C07D217/26; A61K31/4375; A61K31/472; A61K31/4725; A61K31/4741; A61K31/501; A61K31/506; A61K31/5377; A61K31/695; A61P1/04; A61P17/00; A61P19/02; A61P25/00; A61P43/00; C07D401/06; C07D405/06; C07D409/06; C07D413/06; C07D417/06; C07D471/04; C07D491/048; C07D491/056; C07F7/10
Domestic Patent References:
WO2008016659A22008-02-07
WO2004108892A22004-12-16
WO2013042782A12013-03-28
WO2013055984A12013-04-18
WO2013100027A12013-07-04
WO2008121602A12008-10-09
WO2010142752A12010-12-16
Foreign References:
JP2001512137A2001-08-21
Other References:
See also references of EP 3018126A4
"organic synthesis", vol. 22, 1991, article "Jikken Kagaku Kouza", pages: IV
THEODORA W. GREENE; PETER G. M. WUTS: "Protective Groups in Organic Synthesis", 1999, WILEY-INTERSCIENCE, INC.
THEODORA W. GREENE; PETER G. M. WUTS: "Protective Groups in Organic Synthesis", 1999, WILEY-INTERSCIENCE, INC
"Molecule Design", vol. 7, 1990, HIROKAWA SHOTEN, article "Development of Pharmaceutical Products", pages: 163 - 198
JOURNAL OF ANTIBIOTICS, vol. 38, 1985, pages 877 - 885
CHEMICAL AND PHARMACEUTICAL BULLETIN, vol. 38, 1990, pages 2792 - 2796
Attorney, Agent or Firm:
TAKASHIMA, HAJIME (JP)
Takashima 1 (JP)
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