PYRAZOLOPYRIMIDINE-DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS

Title:

PYRAZOLOPYRIMIDINE-DERIVATIVES AS CYCLIN DEPENDENT KINASE INHIBITORS

Document Type and Number:

WIPO Patent Application WO2005077954

Kind Code:

A3

Abstract:

In its many embodiments, the present invention provides pyrazolo[1,5-a]pyrimidine compounds as inhibitors of cyclin dependent kinases, methods of preparing such compounds, pharmaceutical compositions containing one or more such compounds, methods of preparing pharmaceutical formulations comprising one or more such compounds, and methods of treatment, prevention, inhibition, or amelioration of one or more diseases associated with the CDKs using such compounds or pharmaceutical compositions.

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Inventors:

GUZI TIMOTHY J (US)
PARUCH KAMIL (US)
DWYER MICHAEL P (US)
DOLL RONALD J (US)
GIRIJAVALLABHAN VIYYOOR MOOPIL (US)
MALLAMS ALAN (US)
ALVAREZ CARMEN S (US)
KEERTIKAR KARTIK M (US)
RIVERA JOCELYN (US)
CHAN TIN-YAU (US)
MADISON VINCENT (US)
FISCHMANN THIERRY O (US)
DILLARD LAWRENCE W (US)
TRAN VINH D (US)
HE ZHEN MIN (US)
JAMES RAY ANTHONY (US)
PARK HAENGSOON (US)
PARADKAR VIDYADHAR M (US)
HOBBS DOUGLAS WALSH (US)

Application Number:

PCT/US2005/003859

Publication Date:

October 13, 2005

Filing Date:

February 08, 2005

Export Citation:

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Assignee:

SCHERING CORP (US)
PHARMACOPEIA DRUG DISCOVERY (US)
GUZI TIMOTHY J (US)
PARUCH KAMIL (US)
DWYER MICHAEL P (US)
DOLL RONALD J (US)
GIRIJAVALLABHAN VIYYOOR MOOPIL (US)
MALLAMS ALAN (US)
ALVAREZ CARMEN S (US)
KEERTIKAR KARTIK M (US)
RIVERA JOCELYN (US)
CHAN TIN-YAU (US)
MADISON VINCENT (US)
FISCHMANN THIERRY O (US)
DILLARD LAWRENCE W (US)
TRAN VINH D (US)
HE ZHEN MIN (US)
JAMES RAY ANTHONY (US)
PARK HAENGSOON (US)
PARADKAR VIDYADHAR M (US)
HOBBS DOUGLAS WALSH (US)

International Classes:

A61K31/495; C07D487/04; (IPC1-7): C07D487/04; A61K31/495; A61P35/00

Domestic Patent References:

WO1997049378A1	1997-12-31
WO2002050079A1	2002-06-27
WO2004022561A1	2004-03-18
WO2004087707A1	2004-10-14
WO2004022559A1	2004-03-18
WO2004076458A1	2004-09-10

Foreign References:

US6107305A

2000-08-22

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