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Title:
mGluR3の正のアロステリックモジュレーター
Document Type and Number:
Japanese Patent JP6416125
Kind Code:
B2
Abstract:
The present invention relates to novel substituted pyridine derivatives as positive allosteric modulators for modulating metabotropic glutamate receptor subtype 3 (mGluR3) and/or altering glutamate level or glutamatergic signalling.

Inventors:
Justin, Picton
Application Number:
JP2015555607A
Publication Date:
October 31, 2018
Filing Date:
January 22, 2014
Export Citation:
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Assignee:
Plexton Therapeutics Society Anonym
International Classes:
A61K31/5377; A61K31/4365; A61K31/472; A61P1/04; A61P3/00; A61P3/10; A61P7/02; A61P9/10; A61P25/00; A61P25/04; A61P25/06; A61P25/08; A61P25/14; A61P25/16; A61P25/18; A61P25/22; A61P25/24; A61P25/30; A61P27/02; A61P29/00; A61P35/00; A61P43/00
Domestic Patent References:
JP2006512338A
JP2007524710A
JP2009007356A
JP2002521482A
JP2009531370A
JP2006519760A
JP2006511583A
JP2010520876A
JP2009524702A
Foreign References:
EP1074549A1
WO2003093236A1
WO2012085167A1
US6699873
WO2000075101A1
US20070049578
WO2012066077A1
Other References:
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DOUGLAS F. BURDI,JOURNAL OF MEDICINAL CHEMISTRY,2010年10月14日,V53 N19,7107-7118
RAY P.,BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,NL,PERGAMON,2011年 1月 1日,V21 N1,P97-101
Attorney, Agent or Firm:
Kiyoji Kuzuwa