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Title:
METHOD FOR PREPARING 17 alpha-ACETOXY-11beta-(4-N,N-DIMETHYLAMINOPHENYL)-19-NORPREGNA-4,9-DIENE-3,20-DIONE, INTERMEDIATES THEREOF, AND METHODS FOR THE PREPARATION OF SUCH INTERMEDIATES
Document Type and Number:
WIPO Patent Application WO2004078709
Kind Code:
A3
Abstract:
Methods for the preparation of the 19-norprogesterone of formula I and its intermediates, in crystalline and amorphous forms.

Inventors:
KIM HYUN K
RAO PEMMARAJU N
SIMMONS ANNE-MARIE
Application Number:
PCT/US2004/004246
Publication Date:
February 24, 2005
Filing Date:
February 13, 2004
Export Citation:
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Assignee:
US GOV HEALTH & HUMAN SERV (US)
SOUTHWEST FOUND BIOMED RES (US)
KIM HYUN K
RAO PEMMARAJU N
SIMMONS ANNE-MARIE
International Classes:
C07J7/00; C07J21/00; C07D; (IPC1-7): C07J7/00; C07J21/00
Domestic Patent References:
WO2001018025A22001-03-15
Foreign References:
US6020328A2000-02-01
US3381003A1968-04-30
Other References:
See also references of EP 1613640A4
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